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FEMA 4774
CAS No. 1359963-68-0
FEMA 4774( S9632 )
Catalog No. M22734 CAS No. 1359963-68-0
FEMA 4774 is a positive allosteric modulator of T1R2/T1R3.?FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 132 | In Stock |
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| 10MG | 205 | In Stock |
|
| 25MG | 385 | In Stock |
|
| 50MG | 575 | In Stock |
|
| 100MG | 801 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameFEMA 4774
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NoteResearch use only, not for human use.
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Brief DescriptionFEMA 4774 is a positive allosteric modulator of T1R2/T1R3.?FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests.
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DescriptionFEMA 4774 is a positive allosteric modulator of T1R2/T1R3.?FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests.
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In VitroFEMA 4774 (0-50 μM) induces a dose-dependent decrease in the EC50 value of sucrose and significantly enhances the affinity of sucrose for its binding site with an α (effect of modulator on agonist affinity) value of 30 in the human sweet receptor cells.
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In VivoFEMA 4774 (S9632) (oral gavage, 500-2000 mg/kg) does not cause a dose-dependent increase in polychromatic erythrocytes and induces micronuclei formation at dose levels up to 2000 mg/kg in Swiss albino (CD-1) mice.The pharmacokinetic parameters of FEMA 4774 (S9632) in Male and Female Sprague-Dawley Rats.
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SynonymsS9632
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PathwayOthers
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TargetOther Targets
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RecptorT1R2/T1R3
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Research Area——
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Indication——
Chemical Information
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CAS Number1359963-68-0
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Formula Weight359.45
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Molecular FormulaC19H25N3O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 41.67 mg/mL (115.94 )
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SMILESCC(C)NC(=O)C(C)(C)COc1cccc2nc(C)c(C(O)=O)c(N)c12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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